Co Trimoxazole and Warfarin: Drug Interaction Guide
Quick answer: This combination requires caution. Co Trimoxazole and Warfarin can be used together with adjustments and monitoring.
How Co Trimoxazole interacts with Warfarin
Sulfamethoxazole inhibits CYP2C9-mediated metabolism of S-warfarin, while antimicrobial effects on intestinal vitamin K production may further increase INR.
What you should do
Prefer an alternative antibiotic when suitable. If combined, consider warfarin dose adjustment and check INR within several days and again after antibiotic completion.
Key facts
Severity
Moderate — caution required
Mechanism
Sulfamethoxazole inhibits CYP2C9-mediated metabolism of S-warfarin, while antimicrobial effects on intestinal vitamin K ...
Action
Prefer an alternative antibiotic when suitable. If combined, consider warfarin dose adjustment and check INR within seve...
Frequently asked questions
Can I take Co Trimoxazole and Warfarin together?
With caution. Prefer an alternative antibiotic when suitable. If combined, consider warfarin dose adjustment and check INR within several days and again after antibiotic completion.
What is the severity of this interaction?
The interaction between Co Trimoxazole and Warfarin is classified as Moderate — caution required. Sulfamethoxazole inhibits CYP2C9-mediated metabolism of S-warfarin, while antimicrobial effects on intestinal vitamin K production may further increase INR.
What should I do if I'm prescribed both?
Prefer an alternative antibiotic when suitable. If combined, consider warfarin dose adjustment and check INR within several days and again after antibiotic completion. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.