Linezolid and Venlafaxine: Drug Interaction Guide
Quick answer: This is a major interaction — avoid combining Linezolid and Venlafaxine unless specifically directed by your doctor.
How Linezolid interacts with Venlafaxine
Linezolid is a reversible MAO inhibitor; combined with serotonergic SNRIs it can precipitate serotonin syndrome (agitation, hyperthermia, clonus, autonomic instability).
What you should do
Avoid combination. If linezolid is essential, withhold venlafaxine for at least 24 hours before and 2 weeks after linezolid course (5 weeks for fluoxetine).
Key facts
Severity
Major — avoid combination
Mechanism
Linezolid is a reversible MAO inhibitor; combined with serotonergic SNRIs it can precipitate serotonin syndrome (agitati...
Action
Avoid combination. If linezolid is essential, withhold venlafaxine for at least 24 hours before and 2 weeks after linezo...
Frequently asked questions
Can I take Linezolid and Venlafaxine together?
No — this combination should generally be avoided. Avoid combination. If linezolid is essential, withhold venlafaxine for at least 24 hours before and 2 weeks after linezolid course (5 weeks for fluoxetine).
What is the severity of this interaction?
The interaction between Linezolid and Venlafaxine is classified as Major — avoid combination. Linezolid is a reversible MAO inhibitor; combined with serotonergic SNRIs it can precipitate serotonin syndrome (agitation, hyperthermia, clonus, autonomic instability).
What should I do if I'm prescribed both?
Avoid combination. If linezolid is essential, withhold venlafaxine for at least 24 hours before and 2 weeks after linezolid course (5 weeks for fluoxetine). Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.