Erythromycin and Simvastatin: Drug Interaction Guide
Quick answer: This is a major interaction — avoid combining Erythromycin and Simvastatin unless specifically directed by your doctor.
How Erythromycin interacts with Simvastatin
Erythromycin is a strong CYP3A4 inhibitor that markedly increases simvastatin exposure, raising the risk of myopathy and rhabdomyolysis.
What you should do
Withhold simvastatin during the course of erythromycin, or switch to pravastatin or rosuvastatin which are not CYP3A4 substrates.
Key facts
Severity
Major — avoid combination
Mechanism
Erythromycin is a strong CYP3A4 inhibitor that markedly increases simvastatin exposure, raising the risk of myopathy and...
Action
Withhold simvastatin during the course of erythromycin, or switch to pravastatin or rosuvastatin which are not CYP3A4 su...
Frequently asked questions
Can I take Erythromycin and Simvastatin together?
No — this combination should generally be avoided. Withhold simvastatin during the course of erythromycin, or switch to pravastatin or rosuvastatin which are not CYP3A4 substrates.
What is the severity of this interaction?
The interaction between Erythromycin and Simvastatin is classified as Major — avoid combination. Erythromycin is a strong CYP3A4 inhibitor that markedly increases simvastatin exposure, raising the risk of myopathy and rhabdomyolysis.
What should I do if I'm prescribed both?
Withhold simvastatin during the course of erythromycin, or switch to pravastatin or rosuvastatin which are not CYP3A4 substrates. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.